Part of: GH Secretagogues: The Complete GuideTesamorelin doseTesamorelin protocol

Tesamorelin protocol

Tesamorelin dosing — the only FDA-approved GHRH analogue, daily SubQ injection, visceral fat data, off-label body comp use, and side effects.

Updated May 7, 2026 · 5 min read


Tesamorelin is the heavyweight of the GHRH-analogue class. It's the only GH secretagogue with substantial human clinical data behind it, and it's the only one with an FDA approval — for HIV-associated lipodystrophy, sold under the brand name Egrifta. Off-label, it's used for body composition, particularly stubborn visceral fat.

Quick reference

DetailValue
ClassGHRH analogue (modified, longer-acting than Sermorelin)
Half-lifeAbout 30 minutes
CadenceOnce daily
Best timingPre-bed, empty stomach
Typical dose1–2 mg per day
FDA statusApproved for HIV-LD (Egrifta)
Common vials5 mg, 10 mg

Why Tesamorelin is different

Sermorelin, CJC-1295, and Ipamorelin sit in a regulatory gray zone — sold as research chemicals, with limited human trial data outside small studies. Tesamorelin is in a different category. It went through real Phase III clinical trials, received FDA approval, and has a published efficacy and safety record in the population it was studied in.

The clinical record matters for two reasons:

  • Visceral fat reduction is well-documented in the HIV-LD population. The mechanism — GH-axis activation driving lipolysis on visceral adipose — translates to non-HIV users in principle.
  • Side effect profile is better-characterized than other GHRH analogues. You know what you're walking into.

The trade-off: Tesamorelin is more expensive than Sermorelin or CJC-1295, and the side effects are more pronounced because the GH/IGF-1 elevation is meaningfully larger.

Dosing

The FDA-approved dose for HIV-LD is 2 mg SubQ daily. Off-label users typically run 1–2 mg daily depending on tolerance and goals.

GoalDaily dose
Conservative entry1 mg
Standard off-label1.5–2 mg
Approved HIV-LD dose2 mg

Going above 2 mg/day doesn't reliably improve outcomes — the pituitary's release ceiling caps the GH response. Users chasing more effect sometimes split the daily dose into two injections (1 mg morning + 1 mg pre-bed), though most published data is on once-daily pre-bed.

Timing

Pre-bed, empty stomach. Same logic as Sermorelin and Ipamorelin — your largest natural GH pulse occurs in early deep sleep, and the injection amplifies it. High blood glucose blunts the GH response, so eat at least two hours before injection.

The morning option (split dosing) is mostly for users who tolerate Tesamorelin well and want to spread the GH stimulus across the day. There's no strong evidence the split protocol outperforms once-daily pre-bed for body composition.

Reconstitution math

Tesamorelin commonly ships in 5 mg or 10 mg vials. The standard mix:

5 mg vial + 2 mL bacteriostatic water = 2.5 mg/mL.

A 2 mg dose → 0.8 mL → 80 units on a U-100 insulin syringe.

A 1 mg dose → 0.4 mL → 40 units.

For 10 mg vials, doubling to 4 mL BAC water keeps the same concentration. Use the reconstitution calculator for exact units.

Tesamorelin is somewhat more fragile than other GHRH analogues — keep reconstituted vials refrigerated, use within 2–3 weeks, and avoid shaking when mixing.

Cycling

Most off-label users run Tesamorelin in 12–26 week cycles. The visceral fat data shows continued improvement past 26 weeks, but most non-HIV users cycle off to give the GH axis a break and to reset IGF-1 levels.

A common cycle:

PhaseDurationDose
Cycle12–16 weeks1.5–2 mg daily
Off4–8 weeksNone

Bloodwork (IGF-1, fasting glucose, HbA1c) at baseline, mid-cycle, and end-cycle is sensible at this dosage tier. See IGF-1 testing on a GH peptide cycle.

What to expect

Tesamorelin effects build over weeks, not days:

  • Weeks 1–3: improved sleep depth, vivid dreams, mild injection-site reactions
  • Weeks 4–8: subjective recovery improvement, visible body composition shift starts
  • Weeks 9–16: measurable visceral fat reduction, IGF-1 elevation visible on bloodwork

Tesamorelin is not a "feel" drug after each shot. The signal is in the mirror, the waist measurement, and bloodwork at week 12.

Side effects

More pronounced than Sermorelin, generally less than synthetic HGH:

EffectFrequency
Injection-site reactions (redness, irritation)Common
Mild fluid retentionCommon, transient
Joint or muscle achesOccasional
Numbness or tingling in hands or feetOccasional
Mild insulin sensitivity dropCommon at higher doses
HeadacheOccasional

Tesamorelin can shift fasting glucose and insulin sensitivity meaningfully — pre-diabetics and diabetics should be cautious or avoid it. The IGF-1 elevation also raises the same theoretical cancer concerns that apply to all GH-axis interventions; anyone with active or recent cancer should not run Tesamorelin without specialist input.

Deeper coverage: GH secretagogue side effects.

When Tesamorelin makes sense

  • Users who've run Sermorelin or Ipa+CJC and want a stronger GH/IGF-1 signal
  • Users targeting visceral fat specifically (the data is strongest here)
  • Users who value the FDA-backed clinical record over research-chem alternatives

When it doesn't:

  • First-time secretagogue users (start with Sermorelin or Ipa+CJC)
  • Pre-diabetics or diabetics
  • Anyone with active or recent cancer
  • Budget-constrained users (Tesamorelin is the most expensive secretagogue per cycle)
Back to GH Secretagogues: The Complete Guide guide

Related questions

More on gh secretagogues: the complete guide

Free weekly newsletter

Get the strength peptide highlights, weekly.

One short email a week — new guides, study readouts, supply updates, and dosing tips. Plain-English, no spam.

Unsubscribe anytime. We never share your email.